Intengo ye-Medroxyprogesterone Acetate CAS 71-58-9
Incazelo Yomkhiqizo
I-Medroxyprogesterone Acetate, eyaziwa nangokuthi i-Medroxyprogesterone 17-acetate noma i-MPA, iyi-progestogen yokwenziwa kanye ne-steroidal progestin. Itholakala ku-hormone progesterone yomuntu. Ivimbela ukukhulelwa futhi yandisa izinga lokuthuthwa kwamaqanda kusuka kuma-fallopian tubes kuya esibelethweni kuma-ferret abesifazane lapho inikezwa ngaphambi kokuvuthwa. I-Medroxyprogesterone 17-acetate ivimbela ukuvuthwa kwamagundane uma ijovwa ngosuku lokugcina lwe-diestrus. Iphinde ibe nomsebenzi wokulwa ne-androgenic kumagundane, yehlisa amazinga e-testosterone eplasma ngokufakwa komsebenzi we-testosterone reductase yesibindi. I-Medroxyprogesterone 17-acetate ibonisa imiphumela yokucindezela amasosha omzimba ku-vitro kanye naku-vivo, ivimbela ukukhiqizwa kwe-IFN-γ ngamaseli egazi e-CD2/CD3/CD28 ashukunyiswe yi-peripheral blood mononuclear (PBMCs) ngama-concentrations angu-≥10 nM futhi yandisa ukusinda kwama-allografts esikhumba sonogwaja. Izakhi zomjovo eziqukethe i-medroxyprogesterone 17-acetate zisetshenziswe njengezindlela zokuvimbela inzalo.
Ukwenziwa
Isicelo
I-Medroxyprogesterone Acetate iyi-agonist yokwenziwa ye-progesterone receptor esetshenziselwa ukwelapha i-amenorrhea (ukuyeka okungavamile kokuya esikhathini) kanye nokopha okungavamile kwesibeletho.
I-Progestogen:
I-Cachexia (engenalayisensi), ukuvimbela inzalo, isifo sokuwa, ukuxhashazwa kwabesilisa ngokobulili, amathumba abulalayo, izinkinga zokuphefumula, isifo se-sickle-cell, ukopha kwesibeletho okungasebenzi kahle, i-endometriosis.
Ukupakisha Nokugcina Izinto
Ukupakisha: 1 kg/ibhodlela noma 25 kg/isigubhu noma ngokusekelwe ezidingweni zamakhasimende.
Indawo Yokugcina: Gcina endaweni ehlukile, epholile, eyomile futhi enomoya omuhle, futhi uvimbele umswakama ngokuqinile.
Imininingwane
Sicela uthumele i-imeyili ukuze uthole i-COA kanye ne-MSDS.








